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Kerns, RJ
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(1 - 8 of 8)
Title
Suppression of gyrase-mediated resistance by C7 aryl fluoroquinolones
Form
Publication
Date
2016
Collection
Nucleic Acids Research
Title
Selective inhibition of bacterial and human topoisomerase by N-arylacyl O-sulfonated aminoglycoside derivatives
Form
Publication
Date
2013-03-25
Collection
ACS Medicinal Chemistry Letters
Title
Flouroquinolone-gyrase-DNA complexes: two modes or drug binding
Form
Publication
Date
2014-02-04
Collection
Journal of Biological Chemistry
Title
Fluoroquinolones stimulate the DNA cleavage activity of topoisomerase IV by promoting the binding of Mg(2+) to the second metal
Form
Publication
Date
2016-03
Collection
Biochimica et Biophysica Acta
Title
The C-7 aminomethylpyrrolidine group rescues the activity of a thio-fluoroquinolone
Form
Publication
Date
2019-02-11
Collection
Biochimie
Title
Novel N-1 substituted fluoroquinolones inhibit human topoisomerase I activity and exhibit anti-proliferative activity
Form
Publication
Date
2018-09-10
Collection
Investigational New Drugs
Title
Design, synthesis, and evaluation of novel N-1 fluroquinolone derivatives
Form
Publication
Date
2018-06-01
Collection
Bioorg Med Chem Lett
Title
Fluoroquinolones stimulate the DNA cleavage activity of topoisomerase IV
Form
Publication
Date
2016-03
Collection
Biochim Biophys Acta